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Bioactive Compound Library

(4280 compounds) Cat. No.: HY-L001
Library Contents: XLSX PDF

A unique collection of 4280 bioactive compounds including natural products, enzyme inhibitors, receptor ligands, and drugs for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

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Description
& Advantages

•   A unique collection of 4280 bioactive compounds including natural products, enzyme inhibitors, receptor ligands, and drugs for high throughput screening (HTS) and high content screening (HCS).

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some have been approved by FDA.

•   Widely used in the research focus areas such as Cancer, Stem Cell, Neuronal Signaling, Immunity, and more.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and other chemical & biological data.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 4280 bioactive compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Contents of Bioactive Compound Library

Plate layout: HY-L001-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty SKF-96365 (hydrochloride) MRT68921 (hydrochloride) TAK-438 (free base) Ufenamate Calcipotriol CBR-5884 Calcipotriol (monohydrate) Calcitriol HLCL-61 (hydrochloride) Ro 41-1049 (hydrochloride) Empty
b Empty Alfacalcidol PD 117519 YYA-021 Faropenem daloxate Flavopiridol Flavopiridol (Hydrochloride) NPS-2143 SNS-032 Semagacestat Ko 143 Empty
c Empty KNK437 TA-01 AZD-5438 Tubercidin JNJ-17203212 Taranabant PAP-1 4-IBP Toll-like receptor modulator Methoxatin (disodium salt) Empty
d Empty SMER28 HC-067047 EAI045 RSL3 (1S,3R-) IQ-1S (free acid) EPZ015866 Madrasin SZL P1-41 Nutlin (3a) GSK583 Empty
e Empty SRI-011381 (hydrochloride) CL-82198 MS049 DMCM (hydrochloride) MRK-016 (RS)-MCPG E4CPG A 922500 Nigericin (sodium salt) BH3I-1 Empty
f Empty NKL 22 Brevianamide F NVP-BAW2881 F16 PF-04979064 Ro 67-7476 PHCCC FCCP LY2365109 (hydrochloride) Odanacatib Empty
g Empty Imazamox CCF642 HA15 WYE-125132 AEE788 TCS-OX2-29 HO-3867 Plerixafor A-804598 Bay 59-3074 Empty
h Empty TBHQ ITSA-1 Benzophenonetetracarboxylic acid Benzenepentacarboxylic Acid Aprepitant Nanchangmycin Necrosulfonamide Ticagrelor Y-27632 TPCA-1 Empty

Plate layout: HY-L001-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty GMX1778 Triapine Navitoclax Zibotentan LY294002 AS-605240 IC-87114 TG100-115 TGX-221 PI-103 (Hydrochloride) Empty
b Empty Vorapaxar Silodosin AZD1152-HQPA AZD1152 ZM-447439 Veliparib (dihydrochloride) Nilotinib Nilotinib (monohydrochloride monohydrate) Tozasertib Olaparib Empty
c Empty Dabigatran NPS-2143 (hydrochloride) IMD-0354 MLN8054 Dasatinib Dasatinib (hydrochloride) CHIR-99021 Linsitinib NVP-TAE 684 AZD-1480 Empty
d Empty YM-155 SCH 527123 BMS-754807 Sorafenib Sorafenib (Tosylate) Tandutinib OSI-930 Cediranib Amuvatinib Pazopanib Empty
e Empty Masitinib 17-AAG BIIB021 NVP-AUY922 Everolimus Rapamycin Vorinostat CUDC-101 Panobinostat Belinostat Empty
f Empty Bortezomib Motesanib Motesanib (Diphosphate) Saracatinib Telaprevir Boceprevir Danoprevir R-7128 BRAF inhibitor GSK-690693 Empty
g Empty AG1024 PD0325901 Sunitinib SB 203580 SB 203580 (hydrochloride) PD 123319 (ditrifluoroacetate) Vandetanib Afatinib Afatinib (dimaleate) BMS-536924 Empty
h Empty Edoxaban (tosylate monohydrate) Dabigatran etexilate Dabigatran etexilate (mesylate) Linagliptin SB 202190 GSK2126458 GSK-923295 MK-3207 (Hydrochloride) PIK-294 Doramapimod Empty

Plate layout: HY-L001-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty PD173074 BIBX 1382 D4476 CL-387785 GW788388 VX-745 Toceranib Toceranib (phosphate) Regorafenib Regorafenib (monohydrate) Empty
b Empty Brivanib (alaninate) Brivanib Foretinib KW-2449 KX2-391 (dihydrochloride) Fasudil (Hydrochloride) Enzastaurin Sotrastaurin AZD 6482 Raltegravir (potassium salt) Empty
c Empty AKT inhibitor VIII MK 2206 BI-78D3 Canertinib (dihydrochloride) Pim1/AKK1-IN-1 PP121 SU5416 Sutezolid CTS-1027 VX-702 Empty
d Empty Losmapimod SCIO-469 SU 5402 Ki20227 TG-101348 TG101209 MK-2894 AZD-8055 OSI-027 PHA-848125 Empty
e Empty XCT790 SB-431542 A 83-01 SKF-82958 (hydrobromide) HPGDS inhibitor 1 Vismodegib Pralatrexate Capsaicin Dapagliflozin Dapagliflozin ((2S)-1,2-propanediol, hydrate) Empty
f Empty Canagliflozin MLN9708 Carfilzomib TAK-715 PF-562271 (besylate) PF-573228 Daclatasvir (dihydrochloride) Daclatasvir NM107 GSK256066 Empty
g Empty LY2811376 PP 242 AM580 TAK-875 JDTic (dihydrochloride) Dinaciclib Cobicistat BMS-794833 Lexibulin SU14813 Empty
h Empty SU14813 (maleate) Orteronel BI-D1870 AR-A014418 BX795 TSU-68 BMS-345541 BMS-345541 (free base) CGP 57380 Darapladib Empty

Plate layout: HY-L001-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty HIV-1 integrase inhibitor 2 GSK1904529A Telatinib Tasquinimod Betulinic acid GW 5074 Tegobuvir Tariquidar (methanesulfonate, hydrate) RU 58841 Sarpogrelate (hydrochloride) Empty
b Empty Ponesimod Nevirapine Delavirdine (mesylate) Efavirenz Rilpivirine PD 169316 Pluripotin BIO Gatifloxacin Flurbiprofen Empty
c Empty Y-27632 (dihydrochloride) Valproic acid (sodium salt) 5-Azacytidine BIX-01294 TWS119 Neuropathiazol IQ-1 Ro 28-1675 A-966492 Rucaparib (phosphate) Empty
d Empty MK-4827 MK-4827 (tosylate) GW3965 (hydrochloride) LXR-623 SB-705498 AMG 517 Palosuran BMS-687453 MK-6892 PKI-402 Empty
e Empty CJ-42794 EG00229 CCT 137690 Almorexant (hydrochloride) Pemetrexed (disodium) GW 501516 PA-824 Delamanid URB-597 LY2183240 Empty
f Empty Otenabant LRRK2-IN-1 Clotrimazole Istradefylline SB-334867 (free base) SB-674042 TCS 1102 Fexaramine GW2580 UNC0321 Empty
g Empty Aniracetam VER-155008 NVP-BEP800 GNF-7 RG7112 CYT387 CYT387 (sulfate salt) DMXAA SB-590885 Obatoclax Empty
h Empty Alisertib MK-0752 Tivozanib AN-2728 Lenvatinib Amonafide Pomalidomide ENMD-2076 (Tartrate) ENMD-2076 PCI-24781 Empty

Plate layout: HY-L001-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty MGCD-265 analog AZD-7762 MK-1775 Tozadenant PCI-32765 Trametinib Trametinib (DMSO solvate) GSK429286A PHA-793887 CP-466722 Empty
b Empty GW843682X AZ 628 BX-912 KU-57788 GNF-2 CGP60474 TDZD-8 Rivastigmine (tartrate) Risperidone MK-0773 Empty
c Empty WAY-262611 NS11394 Icilin WHI-P97 SB 239063 A-803467 TMC353121 Asenapine (maleate) Alendronate (sodium hydrate) RO4929097 Empty
d Empty Sitaxsentan (sodium) PI3K inhibitor X BIBF 1120 (esylate) PHA-665752 R406 (free base) TAK-242 CGI-1746 AG-490 SNS-314 Fingolimod (hydrochloride) Empty
e Empty Erlotinib (Hydrochloride) Pazopanib (Hydrochloride) BMS-599626 (Hydrochloride) HA14-1 SB 216763 PD153035 (Hydrochloride) SU11274 BSI-201 KU-55933 PF-04217903 Empty
f Empty PF-04217903 (methanesulfonate) Vatalanib SGX-523 INO-1001 Andarine Alvespimycin (hydrochloride) Serdemetan WZ4002 PD98059 PIK-90 Empty
g Empty U0126 2-Methoxyestradiol WYE-354 AMG-208 GSK1059615 Rigosertib (sodium) Ki8751 Elesclomol SP600125 AS703026 Empty
h Empty SB 525334 Cabozantinib (S-malate) HMN-214 PIK-93 Ponatinib Chelerythrine Chloride CCT129202 CP-673451 Vinorelbine (ditartrate) Hesperadin Empty

Plate layout: HY-L001-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty BIX02188 BIX02189 Vemurafenib AT7867 AT7867 (dihydrochloride) KRN-633 KU-60019 PD318088 PHT-427 GSK1292263 Empty
b Empty R406 PI3K-IN-1 SB-743921 DPH LDN193189 LDN193189 (Hydrochloride) Lck Inhibitor LY2109761 BMS 777607 BX471 Empty
c Empty Apremilast Torcetrapib Anacetrapib Oprozomib Poloxin Volasertib A-867744 PNU-120596 Entinostat Mocetinostat Empty
d Empty Aliskiren (hemifumarate) Pitolisant (hydrochloride) TAK-901 PFK-158 PFK-015 RTA-408 PF-06463922 MM-102 (trifluoroacetate) INT-747 PI-3065 Empty
e Empty IWR-1 CID755673 GBR 12935 (dihydrochloride) SB-366791 XEN445 CB-839 T-5224 DMH-1 ML347 FR 180204 Empty
f Empty MI 2 (MALT1 inhibitor) AZ191 K02288 Rostafuroxin MLN1117 PI-1840 YH239-EE Ozanimod Defactinib Arg-Gly-Asp-Ser Empty
g Empty IM-12 PEAQX (tetrasodium hydrate) GKT137831 WH-4-023 MK-3697 Kenpaullone OAC1 IOX1 IBMX Cardiogenol C (hydrochloride) Empty
h Empty Cycloheximide ISX-9 AZD8186 KRCA-0008 HTH-01-015 UNC0379 ML216 ML277 UNC2025 UNC2025 (hydrochloride) Empty

Plate layout: HY-L001-7

1 2 3 4 5 6 7 8 9 10 11 12
a Empty FH1 Ro 61-8048 SB-3CT Siponimod Trenbolone (acetate) C75 (trans) BAY 41-2272 GSK0660 Atipamezole (hydrochloride) Aminothiazole Empty
b Empty SBC-115076 Angiotensin (1-7) 6H05 (trifluoroacetate) PFI-3 G007-LK Y15 SPDB WS6 WS3 A-1210477 Empty
c Empty Decernotinib PF-06447475 BMH-21 LY-2584702 (tosylate salt) LDC1267 ISRIB (trans-isomer) NS-1619 ANA-12 (S)-Willardiine Efonidipine (hydrochloride monoethanolate) Empty
d Empty CFM-2 Pyr6 CX546 Naspm Naspm (trihydrochloride) PEPA SKF-86002 LY3023414 Nicardipine (Hydrochloride) Desogestrel Empty
e Empty OF-1 Oltipraz SKF 38393 (hydrochloride) Bikinin Ro-3306 Dantrolene (sodium hemiheptahydrate) Gonadorelin (acetate) LY3009120 PNU-282987 A-366 Empty
f Empty Thiamet G ZM39923 (hydrochloride) GS967 URMC-099 ON123300 SP2509 Hexachlorophene Dichlorophen Bephenium (hydroxynaphthoate) Pyrantel (pamoate) Empty
g Empty Pyrantel (tartrate) Diethylcarbamazine (citrate) Eprinomectin Acalisib Y16 Primaquine (Diphosphate) Molidustat Entrectinib Glutaminase C-IN-1 BPTES Empty
h Empty CH-223191 Tizoxanide DO3A tert-Butyl ester R(+)-IAA-94 Prucalopride (succinate) 5'-GTP (trisodium salt) 10058-F4 ITD-1 ML324 Liproxstatin-1 Empty

Plate layout: HY-L001-8

1 2 3 4 5 6 7 8 9 10 11 12
a Empty LDN-212320 SCR7 K-7174 (dihydrochloride) AZD3965 ML141 YHO-13177 YHO-13351 (free base) GNE-317 BLZ945 IC261 Empty
b Empty L-779450 Vps34-IN-1 FIPI STF-118804 Optovin EHop-016 TH588 MCC950 MCC950 (sodium) AEBSF Empty
c Empty BLU9931 JNJ-42041935 GSK503 Brigatinib CB-5083 AZD-8835 RBC8 CASIN BQU57 Eliprodil Empty
d Empty Ifenprodil (tartrate) OAC2 PBTZ169 AMG319 ML204 ML204 (hydrochloride) R-268712 Dinoprost (tromethamine salt) Bretylium (tosylate) TP-0903 Empty
e Empty SGI-7079 AZ6102 Spautin-1 Quizartinib Torin 2 Torin 1 PF-3758309 PF-04620110 Laquinimod CH5424802 Empty
f Empty CH5424802 (Hydrochloride) RepSox Cabozantinib Ivacaftor MRT67307 GSK1838705A SRT3190 CC-401 (hydrochloride) DCC-2036 HIV-1 integrase inhibitor Empty
g Empty CAL-101 DAPT (+)-JQ-1 (R)-(-)-JQ1 Enantiomer GSK 525762A CDK-IN-2 LY2784544 R788 (disodium hexahydrate) LX-1031 ADL-5859 Empty
h Empty Cediranib (maleate) Sapitinib LX1606 (Hippurate) SMND-309 ADX-47273 SDZ 220-581 SDZ 220-581 (hydrochloride) IKK-2 inhibitor VIII Daun02 Daunorubicin (Hydrochloride) Empty

Plate layout: HY-L001-9

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Cobimetinib Isobavachalcone Celastrol E-7050 MK-8245 CHIR-98014 MRS 2578 WAY-100635 (maleate salt) CGS 21680 (Hydrochloride) T0070907 Empty
b Empty NVP-TAE 226 Biperiden (Hydrochloride) VX-765 MTEP (hydrochloride) ONX-0914 Ambrisentan Zanamivir (E)-2-Decenoic acid Avasimibe Vanoxerine (dihydrochloride) Empty
c Empty BRL 54443 BAN ORL 24 Crenolanib LY2157299 SD-208 YM-201636 CDK9-IN-1 Rifaximin I-BET151 GSK2578215A Empty
d Empty Dolutegravir (sodium) LY2886721 LY2228820 LY2940680 NXY-059 PF-4136309 GDC-0980 MK-5108 AMG 900 TAME Empty
e Empty OSI-420 Thiazovivin NVP-BHG712 MG-132 CCT128930 A66 VX-809 CHIR-124 WP1130 Droxinostat Empty
f Empty BMS-707035 ABT-751 Tubastatin A (Hydrochloride) Tubastatin-A Dacomitinib JTC-801 IRAK inhibitor 1 IRAK inhibitor 2 IRAK inhibitor 6 PIK-75 Empty
g Empty GANT 58 MF63 Ki16425 SGI-1776 Org 27569 Nepicastat (hydrochloride) KN-62 WIN 55,212-2 (Mesylate) Vinpocetine PYR-41 Empty
h Empty PYZD-4409 Mps1-IN-1 SR-3677 LY2874455 Regorafenib (Hydrochloride) NVP-BGJ398 Montelukast (sodium) Mitomycin C Oseltamivir (acid) JNK-IN-8 Empty

Plate layout: HY-L001-10

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Pracinostat CX-5461 Bardoxolone (methyl) ASP3026 Evacetrapib INK-128 IRAK-1-4 Inhibitor I AZD4547 NVP-BGT226 VU0152100 Empty
b Empty Apatinib ZM 336372 PF-8380 Varespladib INCB28060 SB 242084 Xanomeline (oxalate) AICAR Dorsomorphin (dihydrochloride) U-73122 Empty
c Empty Zebularine SR1001 Zatebradine (hydrochloride) Zatebradine Tenovin-1 RITA FG-4592 (-)-Blebbistatin Nedocromil TAK-733 Empty
d Empty BAY 11-7082 CID 2011756 PHA-767491 (hydrochloride) LY-364947 ALK-IN-1 Debio 0932 GSK126 HG-10-102-01 GNF-5837 ML281 Empty
e Empty Mubritinib Mitoxantrone (dihydrochloride) M344 JNJ-7777120 SA4503 (dihydrochloride) Rupatadine (Fumarate) Camostat (mesylate) U-104 Sirtinol Piceatannol Empty
f Empty TRAM-34 Nocodazole SB-505124 PAC-1 AG-1478 LY310762 CAY10505 AS-252424 AZD-2461 Gemcitabine (elaidate) Empty
g Empty Exherin (trifluoroacetate) Uramustine Amsacrine Anidulafungin β-Lapachone Ascomycin AZM475271 Betamethasone Beclometasone dipropionate Biapenem Empty
h Empty Blonanserin BTZ043 Budesonide Carmustine Cefsulodin (sodium) Chlorambucil Cisatracurium (besylate) Cladribine Clobetasol propionate Cyproterone (acetate) Empty

Plate layout: HY-L001-11

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Cytarabine Dacinostat Deflazacort Dutasteride Efaproxiral Efaproxiral (sodium) Entecavir (monohydrate) Epirubicin (hydrochloride) Estramustine (phosphate sodium) Etoposide Empty
b Empty Exemestane Ezatiostat Finasteride Fulvestrant Ganciclovir GDC-0152 RG108 Daminozide (-)-Epigallocatechin Gallate Lansoprazole Empty
c Empty (R)-Lansoprazole Folinic acid (Calcium) Levamisole (hydrochloride) Levoleucovorin (Calcium) Lomeguatrib Lomustine Megestrol (Acetate) 6-Mercaptopurine Meropenem (trihydrate) Mesna Empty
d Empty Mifepristone Miltefosine PQ401 IKK 16 PJ34 (hydrochloride) Mitotane Mometasone furoate MSX-122 Nandrolone decanoate Nedaplatin Empty
e Empty Nelarabine SN-38 Norepinephrine (bitartrate monohydrate) Noscapine