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  2. Metabolism/Protease Compound Library

Metabolism/Protease Compound Library

(797 compounds) Cat. No.: HY-L012
Library Contents: XLSX PDF

A unique collection of 797 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

  • Documentation

& Advantages

•   A unique collection of 797 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as PDE, Cytochrome P450, HMG-CoA Reductase, DPP4, Proteasome, HCV Protease, IDO, Cathepsin, MMP, etc.

•   A useful tool for drug discovery of metabolism-related diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
A collection of 797 Metabolism/Protease related compounds supplied as pre-dissolved DMSO solutions or Solid
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Blue ice

Contents of Metabolism/Protease Compound Library

Plate layout: HY-L012-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty KNK437 CL-82198 A 922500 Odanacatib GMX1778 Dabigatran 17-AAG BIIB021 NVP-AUY922 Bortezomib Empty
b Empty Telaprevir Boceprevir Danoprevir Edoxaban (tosylate monohydrate) Dabigatran etexilate Dabigatran etexilate (mesylate) Linagliptin Raltegravir (potassium salt) CTS-1027 MLN9708 Empty
c Empty Carfilzomib Daclatasvir (dihydrochloride) Daclatasvir GSK256066 Cobicistat Orteronel HIV-1 integrase inhibitor 2 Ro 28-1675 URB-597 LY2183240 Empty
d Empty VER-155008 NVP-BEP800 AN-2728 Alvespimycin (hydrochloride) 2-Methoxyestradiol Apremilast Oprozomib Aliskiren (hemifumarate) PI-1840 IBMX Empty
e Empty SB-3CT Oltipraz Molidustat STF-118804 AEBSF JNJ-42041935 PF-04620110 HIV-1 integrase inhibitor LX-1031 LX1606 (Hippurate) Empty
f Empty Celastrol MK-8245 ONX-0914 Dolutegravir (sodium) MG-132 BMS-707035 Nepicastat (hydrochloride) Vinpocetine PF-8380 U-73122 Empty
g Empty FG-4592 Debio 0932 β-Lapachone Cladribine Dutasteride Finasteride Sitagliptin Sitagliptin (phosphate monohydrate) NLG919 Zileuton Empty
h Empty Milrinone Olprinone (Hydrochloride) Febuxostat Anastrozole Vildagliptin PF-04457845 PF-3845 AT13387 Talarozole Lopinavir Empty

Plate layout: HY-L012-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Biochanin A Fluvastatin (sodium) Elvitegravir Teneligliptin Teneligliptin (hydrobromide) Anagliptin Bay 60-7550 Sildenafil (citrate) Balicatib Lonafarnib Empty
b Empty Oglemilast NVP-HSP990 Ganetespib Geldanamycin JZL 184 JZL195 Tiplaxtinin E-64 Nelfinavir (Mesylate) Trelagliptin Empty
c Empty Trelagliptin (succinate) CPI-613 Roflumilast IOX2 Cabotegravir Alvelestat IDO5L INCB 024360 PluriSln 1 AGI-6780 Empty
d Empty GM6001 NSC 405020 FTI-277 (hydrochloride) DMOG P7C3 Tolrestat Dafadine-A Indoximod Rolipram (R)-(-)-Rolipram Empty
e Empty SW033291 Saquinavir (Mesylate) Saquinavir Darunavir (Ethanolate) Atazanavir (sulfate) Dabigatran (ethyl ester) Atorvastatin (hemicalcium salt) Mevastatin Amprenavir Sivelestat (sodium tetrahydrate) Empty
f Empty Cilostazol Simvastatin Rosuvastatin (Calcium) Clarithromycin Daprodustat AGI-5198 Lisinopril (dihydrate) Leupeptin (hemisulfate) Avanafil Udenafil Empty
g Empty PU-WS13 Enasidenib VR23 Ivosidenib (R,S)-Ivosidenib KC7F2 Alda-1 Aldose reductase-IN-1 KML29 HA130 Empty
h Empty DASA-58 TMS JNJ-42165279 PD 151746 Methoxsalen T863 Etomoxir (R)-(+)-Etomoxir (sodium salt) Apixaban DGAT-1 inhibitor 2 Empty

Plate layout: HY-L012-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty A939572 FK866 Rivaroxaban Epalrestat Carboxypeptidase G2 (CPG2) Inhibitor CPA inhibitor TOK-001 Abiraterone Otamixaban GSK256066 (2,2,2-trifluoroacetic acid) Empty
b Empty Abiraterone (acetate) DMP 777 FAAH-IN-2 Ritonavir Nortadalafil Tadalafil Pentostatin Alogliptin (Benzoate) Cilazapril (monohydrate) Malotilate Empty
c Empty Diphylline Perindopril (erbumine) Aminophylline Pitavastatin (Calcium) Pravastatin (sodium) Nafamostat (mesylate) Pimobendan Allopurinol Enalaprilat (dihydrate) Disulfiram Empty
d Empty Ramipril Dipyridamole Enalapril (maleate) Captopril Argatroban (monohydrate) Moexipril (hydrochloride) Fosinopril (sodium) Temocapril (hydrochloride) Gabexate (mesylate) Ozagrel Empty
e Empty Ozagrel (sodium) Vardenafil (hydrochloride) Quinapril (hydrochloride) PMSF Anagrelide (hydrochloride) Zofenopril (calcium) Indinavir (sulfate) Pentoxifylline Ibudilast Teprenone Empty
f Empty Theophylline Benzbromarone Metyrapone Proadifen (hydrochloride) Imidapril (hydrochloride) Chlorzoxazone Carbosulfan 3-Cyano-7-ethoxycoumarin Chlorogenic acid Isoliquiritigenin Empty
g Empty Naringin Lovastatin Pepstatin Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

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